
Preclinical characterization and first-in-human administration of a selective monoacylglycerol lipase inhibitor, ABX-1431
Author(s) -
Iain D. C. Fraser,
Jacqueline L. Blankman,
Jason R. Clapper,
Cheryl A. Grice,
Gary P. O’Neill,
Alan Ezekowitz,
Archie W. Thurston,
Els Geenens,
Corinne Vandermeulen,
Jan de Hoon
Publication year - 2017
Publication title -
frontiers in pharmacology
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 1.384
H-Index - 86
ISSN - 1663-9812
DOI - 10.3389/conf.fphar.2017.62.00011
Subject(s) - monoacylglycerol lipase , pharmacology , endocannabinoid system , peripheral blood mononuclear cell , lipase , biology , medicine , chemistry , enzyme , receptor , biochemistry , in vitro