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THE INTERACTION OF NICOTINIC RECEPTOR ANTAGONISTS AT MUSCARINIC RECEPTORS
Author(s) -
Mitchelson F. J.
Publication year - 1987
Publication title -
clinical and experimental pharmacology and physiology
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 0.752
H-Index - 103
eISSN - 1440-1681
pISSN - 0305-1870
DOI - 10.1111/j.1440-1681.1987.tb00988.x
Subject(s) - muscarinic acetylcholine receptor , nicotinic agonist , pharmacology , receptor , muscarinic acetylcholine receptor m3 , muscarinic acetylcholine receptor m2 , alpha 4 beta 2 nicotinic receptor , chemistry , muscarinic acetylcholine receptor m1 , muscarinic acetylcholine receptor m4 , medicine , neuroscience , psychology , nicotinic acetylcholine receptor
SUMMARY 1. The interaction of some neuromuscular blocking drugs such as gallamine, pancuronium and stercuronium with muscarinic receptors has several features which distinguish these compounds from competitive antagonists in functional and binding studies. 2. They also differentiate between muscarinic receptors and may produce effects on ion channels.

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