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GABA B receptors in the bladder and bowel: therapeutic potential for positive allosteric modulators?: Commentary on Kalinichev et al ., Br J Pharmacol 171: 995–1006
Author(s) -
Hyland Niall P,
Golubeva Anna V
Publication year - 2015
Publication title -
british journal of pharmacology
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 2.432
H-Index - 211
eISSN - 1476-5381
pISSN - 0007-1188
DOI - 10.1111/bph.12617
Subject(s) - allosteric regulation , receptor , pharmacology , neuroscience , medicine , gabaa receptor , allosteric modulator , chemistry , biology
Linked Article This article is a Commentary on Kalinichev M, Palea S, Haddouk H, Royer‐Urios I, Guilloteau V, Lluel P, Schneider M, Saporito M and Poli S (2014). ADX71441, a novel, potent and selective positive allosteric modulator of the GABAB receptor, shows efficacy in rodent models of overactive bladder. Br J Pharmacol 171: 995–1006. doi: 10.1111/bph.12517