Structure-based design of haloperidol analogues as inhibitors of acetyltransferase Eis from Mycobacterium tuberculosis to overcome kanamycin resistance
Author(s) -
Ankita Punetha,
Keith Green,
Atefeh Garzan,
Nishad Thamban Chandrika,
Melisa J. Willby,
Allan H. Pang,
Caixia Hou,
Selina Y. L. Holbrook,
Kyle Krieger,
James E. Posey,
Tanya Parish,
Oleg V. Tsodikov,
Sylvie GarneauTsodikova
Publication year - 2021
Publication title -
rsc medicinal chemistry
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 0.754
H-Index - 55
ISSN - 2632-8682
DOI - 10.1039/d1md00239b
Subject(s) - haloperidol , pharmacology , chemistry , mycobacterium tuberculosis , antipsychotic , medicine , tuberculosis , dopamine , schizophrenia (object oriented programming) , pathology , psychiatry
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