Discovery and Lead Optimization of Benzene-1,4-disulfonamides as Oxidative Phosphorylation Inhibitors
Author(s) -
Ding Xue,
Yibin Xu,
Armita Kyani,
Joyeeta Roy,
Lipeng Dai,
Duxin Sun,
Nouri Neamati
Publication year - 2022
Publication title -
journal of medicinal chemistry
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 2.01
H-Index - 261
eISSN - 1520-4804
pISSN - 0022-2623
DOI - 10.1021/acs.jmedchem.1c01509
Subject(s) - chemistry , oxidative phosphorylation , cytotoxicity , biochemistry , adenosine triphosphate , phosphorylation , structure–activity relationship , pancreatic cancer , lead compound , pharmacology , combinatorial chemistry , in vitro , cancer , biology , genetics
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