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High specific activity tritium labeling of anti‐tumor agent CEP‐2563
Author(s) -
Egan Judith A.,
Filer Crist N.,
Hudkins Robert L.
Publication year - 2005
Publication title -
journal of labelled compounds and radiopharmaceuticals
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 0.432
H-Index - 47
eISSN - 1099-1344
pISSN - 0362-4803
DOI - 10.1002/jlcr.1010
Subject(s) - chemistry , tritium , tritium illumination , radiochemistry , specific activity , combinatorial chemistry , biochemistry , enzyme , nuclear physics , physics
Abstract [Ester Methylene‐ 3 H] CEP‐2563 ( 9 ) was synthesized by the tritiation of precursor 6 with NaB 3 H 4 followed by esterification with BOC‐Lys(BOC)‐ β ‐Ala‐OH and deprotection. Copyright © 2005 John Wiley & Sons, Ltd.