Preparation and reactivity of 5‐substituted azepino[3,4‐ b ]indoles | Zendy

Montagne C. | Zendy; Laurent N. | Zendy; Joseph B. | Zendy; Mérour J.Y. | Zendy

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Preparation and reactivity of 5‐substituted azepino[3,4‐ b ]indoles

Author(s) -

Montagne C.,

Laurent N.,

Joseph B.,

Mérour J.Y.

Publication year - 2005

Publication title -

journal of heterocyclic chemistry

Language(s) - English

Resource type - Journals

SCImago Journal Rank - 0.321

H-Index - 59

eISSN - 1943-5193

pISSN - 0022-152X

DOI - 10.1002/jhet.5570420728

Subject(s) - indole test , chemistry , reactivity (psychology) , scope (computer science) , catalysis , combinatorial chemistry , heck reaction , medicinal chemistry , organic chemistry , stereochemistry , palladium , medicine , alternative medicine , pathology , computer science , programming language

Preparation of the 5‐substituted azepino[3,4‐ b ]indole core structure can be realised through a catalytic Heck reaction. The scope and limitations of this methodology are reported. The reactivity of di‐ tert ‐butyl 5‐ethoxycarbonylmethylene‐1,3,4,5‐tetrahydro‐1‐oxoazepino[3,4‐b]indole‐2,10‐dicarboxylate (1) was investigated in order to prepare the indole analogue of hymenialdisine and derivatives.

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