Premium
2‐Azidopyrrolo[2,1‐ c ][1,4]benzodiazepines. Synthesis of the first cyclic amidine derivatives
Author(s) -
Gillard AlainClaude,
Rault Sylvain
Publication year - 1997
Publication title -
journal of heterocyclic chemistry
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 0.321
H-Index - 59
eISSN - 1943-5193
pISSN - 0022-152X
DOI - 10.1002/jhet.5570340415
Subject(s) - chemistry , amidine , benzazepines , medicinal chemistry , stereochemistry , organic chemistry
Abstract We report the practical synthesis of the new 5‐azidopyrrolo[2,1‐ c ][1,2,4]triazolo[4,3‐ a ][1,4]benzo‐diazepin‐8‐one and 11‐alkylamino‐2‐azidopyrrolo[2,1‐ c ][1,4]benzodiazepines via the corresponding hydroxy compounds.