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Synthesis of [1,2,4]triazoloquinazoline and [1,2,4]‐triazolo‐1,4‐benzodiazepine derivatives
Author(s) -
Gatta Franco,
Del Giudice Maria Rosaria,
Borioni Anna
Publication year - 1993
Publication title -
journal of heterocyclic chemistry
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 0.321
H-Index - 59
eISSN - 1943-5193
pISSN - 0022-152X
DOI - 10.1002/jhet.5570300102
Subject(s) - chemistry , d 1 , benzodiazepine , stereochemistry , biochemistry , receptor
Some [1,2,4]triazolo[1,5‐ c ]quinazolin‐5(6 H )‐ones 7 , the corresponding isomers [1,2,4]triazolo[4,3‐ c ]quinazo‐lin‐5(6 H )‐ones and the 5‐amino derivatives 8, 9 and 11 have been synthesized starting from the acylamidrazones 5 . The preparation of 5 H ‐[1,2,4]triazolo[1,5‐ d ]‐1,4‐benzodiazepin‐6(7 H )‐ones 15 and of 5‐cyclicaminomethyl‐[1,2,4]triazolo[1,5‐ c ]quinazolines 16 and 17 is also reported.