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A facile synthesis of 3‐amino‐5‐substitutedaminoisothiazole‐4‐carboxylic acid derivatives
Author(s) -
Shishoo C. J.,
Devani M. B.,
Ananthan S.,
Bhadti V. S.,
Ullas G. V.
Publication year - 1988
Publication title -
journal of heterocyclic chemistry
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 0.321
H-Index - 59
eISSN - 1943-5193
pISSN - 0022-152X
DOI - 10.1002/jhet.5570250311
Subject(s) - chemistry , carboxylic acid , organic chemistry , combinatorial chemistry
A facile, general and one‐pot method for the preparation of 3‐amino‐5‐substituted‐aminoisothiazole‐4‐carboxylic acid derivatives, in high yields, by the aminative cyclization of 3‐amino‐3‐mercaptoacrylonitriles is described.