Synthesis of 3 H [1,2]diazepino[5,6‐ b ]indole and 3 H [1,2]diazepino[4,5‐ b ]indole derivatives | Zendy

Monge A. | Zendy; Palop J. A. | Zendy; Goñi T. | Zendy; Martinez A. | Zendy; FernándezAlvarez E. | Zendy

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Synthesis of 3 H [1,2]diazepino[5,6‐ b ]indole and 3 H [1,2]diazepino[4,5‐ b ]indole derivatives

Author(s) -

Monge A.,

Palop J. A.,

Goñi T.,

Martinez A.,

FernándezAlvarez E.

Publication year - 1984

Publication title -

journal of heterocyclic chemistry

Language(s) - English

Resource type - Journals

SCImago Journal Rank - 0.321

H-Index - 59

eISSN - 1943-5193

pISSN - 0022-152X

DOI - 10.1002/jhet.5570210221

Subject(s) - chemistry , hydrazine (antidepressant) , indole test , formylation , acetonitrile , derivative (finance) , medicinal chemistry , organic chemistry , stereochemistry , catalysis , chromatography , financial economics , economics

The synthesis of two new derivatives of 3 H [1,2]diazepino[5,6‐ b ]indole, 5 and 11 , and one new derivative of 3 H [1,2]diazepino[4,5‐ b ]indole, 16 , are described. Compound 5 was obtained by the reaction of methyl 2‐(3‐methoxycarbonyl‐1‐methylindole)acetate 2 , with hydrazine. Compound 11 was obtained in two ways from ethyl 2‐(1‐methylindole)acetate ( 8 ) by formylation and reaction with hydrazine. Compound 16 was obtained treating 3‐(2‐ethoxycarbonylindole)acetonitrile ( 14 ) with hydrazine.

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