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Syntheses of 2‐arylimidazole derivatives through annelations employing benzylamines
Author(s) -
Veronese A. C.,
Cavicchioni G.,
Servadio G.,
Vecchiati G.
Publication year - 1980
Publication title -
journal of heterocyclic chemistry
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 0.321
H-Index - 59
eISSN - 1943-5193
pISSN - 0022-152X
DOI - 10.1002/jhet.5570170816
Subject(s) - chemistry , imidazole , alkyl , organic chemistry , pentane , combinatorial chemistry
Annelations of benzylamines with hydroximino derivatives of pentane‐2,4‐dione or of alkyl acetoacetates, acetoacetamides, and acetoacetanilides, afford imidazole derivatives and provide easy incorporation of the benzylic carbon and nitrogen in the heterocycle. The limits of the reaction have been explored.