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Fused indoles. 1. Synthesis of the 1,9‐dihydrothiazino[3,4‐ b ] indole ring system
Author(s) -
Coppola Gary M.,
Hardtmann Goetz E.
Publication year - 1977
Publication title -
journal of heterocyclic chemistry
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 0.321
H-Index - 59
eISSN - 1943-5193
pISSN - 0022-152X
DOI - 10.1002/jhet.5570140640
Subject(s) - chemistry , indole test , sodium hydride , ring (chemistry) , medicinal chemistry , sodium , spectral properties , hydride , stereochemistry , combinatorial chemistry , organic chemistry , computational chemistry , hydrogen
The title compounds were prepared by treating 2‐chloroindole‐3‐carboxaldehydes and 3‐acetyl‐2‐chloroindole with N ‐methylmethanesulfonamide and cyclizing the resulting intermediates with sodium hydride. Spectral data of the products are also discussed. J. Chem. Soc. , 14, 1117 (1977)