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Psilocin analogs. 1. Synthesis of 3‐[2‐(dialkylamino)ethyl] ‐and 3‐[2‐(cycloalkylamino)ethyl] indol‐4‐ols
Author(s) -
Repke David B.,
Ferguson Wilfred J.,
Bates Dallas K.
Publication year - 1977
Publication title -
journal of heterocyclic chemistry
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 0.321
H-Index - 59
eISSN - 1943-5193
pISSN - 0022-152X
DOI - 10.1002/jhet.5570140113
Subject(s) - chemistry , stereochemistry , combinatorial chemistry
The synthesis of four dialkyl and three eyeloalkyl analogs of psilocin (4, R ‐ CH 3 ), a hallucinogenic principle found in certain fungi, is described. The synthetic route involves four transformations starting with 6,7‐dihydroindol‐4(5 H )one: (1).
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