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Diastereodivergent Synthesis of Pyrazoline Derivatives through [3 + 2] Cycloaddition of Baylis–Hillman Adducts and Nitrilimines
Author(s) -
Zeng Yuan,
Zhou Leijie,
Gao Xing,
Wu Yang,
Wang Qijun,
Guo Zhenyan,
Huang Jiaxing,
Guo Hongchao
Publication year - 2018
Publication title -
journal of heterocyclic chemistry
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 0.321
H-Index - 59
eISSN - 1943-5193
pISSN - 0022-152X
DOI - 10.1002/jhet.3344
Subject(s) - chemistry , cycloaddition , adduct , pyrazoline , combinatorial chemistry , medicinal chemistry , organic chemistry , catalysis
In this paper, a [3 + 2] cycloaddition of Baylis–Hillman adducts and nitrilimines has been achieved under mild reaction conditions, providing a concise approach to access biologically important pyrazoline derivatives.