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Design, Synthesis, and Biological Screening of Novel Anthranilic Diamides
Author(s) -
Hua Xuewen,
Mao Wutao,
Fan Zhijin,
Ji Xiaotian,
Li Fengyun,
Zong Guangning,
Song Haibin,
Tatiana Kalinina,
Morzherin Yury Yu.,
Belskaya Nataliya P.,
Bakulev Vasiliy A.
Publication year - 2016
Publication title -
journal of heterocyclic chemistry
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 0.321
H-Index - 59
eISSN - 1943-5193
pISSN - 0022-152X
DOI - 10.1002/jhet.2351
Subject(s) - chemistry , mythimna separata , sclerotinia sclerotiorum , anthranilic acid , elemental analysis , proton nmr , fungicide , organic chemistry , stereochemistry , botany , lepidoptera genitalia , biology
Three series of new anthranilic diamide derivatives containing sulfide, N ‐cyanomethylsulfilimine, and N ‐cyanomethylsulfoximine groups were designed and synthesized by combining the active substructures of anthranilic diamides and sulfoxaflor. The structures of all newly synthesized compounds were confirmed by IR and 1 H/ 13 C‐NMR, and some of them were confirmed by elemental analysis or HRMS too. The synthesized compounds were screened for their insecticidal and fungicidal activities. Bioasssay results indicated that some of the synthesized compounds possessed certain degrees of insecticidal activity against Mythimna separata . However, some compounds exhibited good fungicidal activity against Sclerotinia sclerotiorum .