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The Synthesis of Some 7, 8‐Dimethoxy‐5‐phenyl‐2 H ‐3‐benzazepin‐2‐one Derivatives
Author(s) -
Berney Daniel,
Schuh Karlheinz
Publication year - 1981
Publication title -
helvetica chimica acta
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 0.74
H-Index - 82
eISSN - 1522-2675
pISSN - 0018-019X
DOI - 10.1002/hlca.19810640202
Subject(s) - chemistry , benzazepine , chloride , stereochemistry , combinatorial chemistry , medicinal chemistry , organic chemistry
The benzazepin‐2‐ones 7 and 9 were prepared from homoveratroyl chloride (4) and phenacylamine. Compounds 7 and 9 were used for the preparation of the benzazepin‐2‐amines 3, 11, 13 and 14. A synthesis of the benzazepine‐1,2‐dione 17 and the benzazepine‐2,4‐dione 20 is also described.