Convenient Synthesis of Thieno[3,2‐ b ]indoles and Thieno[3,4‐ b ]indoles by Sequential Site‐Selective Suzuki and Double C–N Coupling Reactions | Zendy

Pham Ngo Nghia | Zendy; Parpart Silvio | Zendy; Grigoryan Sevak | Zendy; Ngo Thang Ngoc | Zendy; Dang Tuan Thanh | Zendy; Ghochikyan Tariel V. | Zendy; Saghyan Ashot S. | Zendy; Ehlers Peter | Zendy; Langer Peter | Zendy

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Convenient Synthesis of Thieno[3,2‐ b ]indoles and Thieno[3,4‐ b ]indoles by Sequential Site‐Selective Suzuki and Double C–N Coupling Reactions

Author(s) -

Pham Ngo Nghia,

Parpart Silvio,

Grigoryan Sevak,

Ngo Thang Ngoc,

Dang Tuan Thanh,

Ghochikyan Tariel V.,

Saghyan Ashot S.,

Ehlers Peter,

Langer Peter

Publication year - 2017

Publication title -

european journal of organic chemistry

Language(s) - English

Resource type - Journals

SCImago Journal Rank - 0.825

H-Index - 155

eISSN - 1099-0690

pISSN - 1434-193X

DOI - 10.1002/ejoc.201601281

Subject(s) - chemistry , suzuki reaction , stereochemistry , combinatorial chemistry , coupling reaction , indole test , organic chemistry , palladium , catalysis

A convenient synthesis of thieno[3,2‐ b ]indoles and thieno[3,4‐ b ]indoles has been developed. The protocol involves a site‐selective Suzuki reaction, followed by a double C–N coupling reaction using anilines, benzylamines, or alkylamines. The yields range from good to excellent.

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