Access to Imidazo[1,2‐ a ]imidazolin‐2‐ones and Functionalization through Suzuki–Miyaura Cross‐Coupling Reactions | Zendy

Grosse Sandrine | Zendy; Pillard Christelle | Zendy; Himbert Franck | Zendy; Massip Stéphane | Zendy; Léger Jean Michel | Zendy; Jarry Christian | Zendy; Bernard Philippe | Zendy; Guillaumet Gérald | Zendy

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Access to Imidazo[1,2‐ a ]imidazolin‐2‐ones and Functionalization through Suzuki–Miyaura Cross‐Coupling Reactions

Author(s) -

Grosse Sandrine,

Pillard Christelle,

Himbert Franck,

Massip Stéphane,

Léger Jean Michel,

Jarry Christian,

Bernard Philippe,

Guillaumet Gérald

Publication year - 2013

Publication title -

european journal of organic chemistry

Language(s) - English

Resource type - Journals

SCImago Journal Rank - 0.825

H-Index - 155

eISSN - 1099-0690

pISSN - 1434-193X

DOI - 10.1002/ejoc.201300268

Subject(s) - chemistry , combinatorial chemistry , bromine , aryl , surface modification , coupling reaction , boronic acid , organic chemistry , catalysis , alkyl

We report herein a synthetic pathway to new 6(5)‐bromo‐5(6)‐methylimidazo[1,2‐ a ]imidazolin‐2‐ones. The synthetic potential of these scaffolds was demonstrated by displacing bromine by Suzuki–Miyaura cross‐coupling reactions. A large panel of boronic acids (aryl, heteroaryl or vinyl) could easily be introduced, giving access to a large and diversified library of 6(5)‐substituted 5(6)‐methylimidazo[1,2‐ a ]imidazolin‐2‐ones.

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