Diversely Substituted Triazolo[1,5‐ a ][1,4]benzodiazepinones: A Post‐Ugi Copper‐Catalyzed Tandem Azide–Alkyne Cycloaddition/Ullmann C–N Coupling Approach | Zendy

Vachhani Dipak D. | Zendy; Kumar Amit | Zendy; Modha Sachin G. | Zendy; Sharma Sunil K. | Zendy; Parmar Virinder S. | Zendy; Van der Eycken Erik V. | Zendy

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Diversely Substituted Triazolo[1,5‐ a ][1,4]benzodiazepinones: A Post‐Ugi Copper‐Catalyzed Tandem Azide–Alkyne Cycloaddition/Ullmann C–N Coupling Approach

Author(s) -

Vachhani Dipak D.,

Kumar Amit,

Modha Sachin G.,

Sharma Sunil K.,

Parmar Virinder S.,

Van der Eycken Erik V.

Publication year - 2013

Publication title -

european journal of organic chemistry

Language(s) - English

Resource type - Journals

SCImago Journal Rank - 0.825

H-Index - 155

eISSN - 1099-0690

pISSN - 1434-193X

DOI - 10.1002/ejoc.201201587

Subject(s) - cycloaddition , chemistry , alkyne , tandem , azide , catalysis , copper , combinatorial chemistry , stereochemistry , organic chemistry , materials science , composite material

A diversity‐oriented approach comprising an Ugi 4‐component reaction and a copper‐catalyzed tandem azide–alkyne cycloaddition/Ullmann C–N coupling is elaborated. The methodology is compatible with various functional groups and allows the construction of triazolo[1,5‐ a ][1,4]benzodiazepinones in good yields.

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