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3‐(Arylamino)‐1,2,4‐triazin‐5‐one: A Novel Synthesis and Its Use
Author(s) -
Leenders Ruben,
Heeres Jan,
Vandenput Dirk,
Zijlmans Remco,
Guillemont Jérôme,
Lewi Paul
Publication year - 2010
Publication title -
european journal of organic chemistry
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 0.825
H-Index - 155
eISSN - 1099-0690
pISSN - 1434-193X
DOI - 10.1002/ejoc.201000242
Subject(s) - chemistry , triazine , combinatorial chemistry , surface modification , core (optical fiber) , protocol (science) , position (finance) , nanotechnology , organic chemistry , computer science , telecommunications , medicine , alternative medicine , pathology , finance , economics , materials science
An optimized procedure is given for the synthesis of novel 3‐(arylamino)‐1,2,4‐triazin‐5‐one building blocks from commercially available material. By employing these building blocks, a practical protocol is described for the functionalization of the 5‐position of the triazine core with anilines orphenols.