Copper(I)‐Catalyzed Cascade Synthesis of 2‐Substituted 1,3‐Benzothiazoles: Direct Access to Benzothiazolones | Zendy

Murru Siva | Zendy; Mondal Pravat | Zendy; Yella Ramesh | Zendy; Patel Bhisma K. | Zendy

AI Assistant Blog Pricing

Home ZAIA Blog

Premium

Copper(I)‐Catalyzed Cascade Synthesis of 2‐Substituted 1,3‐Benzothiazoles: Direct Access to Benzothiazolones

Author(s) -

Murru Siva,

Mondal Pravat,

Yella Ramesh,

Patel Bhisma K.

Publication year - 2009

Publication title -

european journal of organic chemistry

Language(s) - English

Resource type - Journals

SCImago Journal Rank - 0.825

H-Index - 155

eISSN - 1099-0690

pISSN - 1434-193X

DOI - 10.1002/ejoc.200900711

Subject(s) - chemistry , intramolecular force , cascade , catalysis , alkyl , combinatorial chemistry , nucleophile , medicinal chemistry , stereochemistry , organic chemistry , chromatography

An efficient cascade process for the preparation of 2‐substituted 1,3‐benzothiazoles directly from 2‐haloaryl isothiocyanates and O or S nucleophiles by a Cu‐catalyzed, intramolecular, C–S bond formation has been developed. This cascade method is viable for the efficient syntheses of both O‐ and S‐substituted 1,3‐benzothiazoles. Furthermore, 1,3‐benzothiazol‐2(3 H )‐ones having an alkyl group allow easy access to 1,3‐benzothiazolones. (© Wiley‐VCH Verlag GmbH & Co. KGaA, 69451 Weinheim, Germany, 2009)

This content is not available in your region!

Continue researching here.

Having issues? You can contact us here

Accelerating Research