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An Improved Protocol for Regioselective Ring‐Opening of Sulfonyl Aziridines with Iodine Promoted by PPh 3
Author(s) -
Zhang Jinfeng,
Meng Lingguo,
Li Chuntao,
Xiao Guoyuan
Publication year - 2013
Publication title -
chinese journal of chemistry
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 1.28
H-Index - 41
eISSN - 1614-7065
pISSN - 1001-604X
DOI - 10.1002/cjoc.201300625
Subject(s) - chemistry , chemoselectivity , sulfonyl , regioselectivity , iodine , ring (chemistry) , combinatorial chemistry , reaction conditions , organic chemistry , medicinal chemistry , catalysis , alkyl
A new route to synthesize β ‐iodo amines from sulfonyl aziridines and iodine was developed in the presence of PPh 3 . This ring‐opening reaction was an efficient and simple process to give β ‐iodo amines in excellent yields with high chemoselectivity.