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Synthesis and Bioactivities of Novel N ‐(4‐(2‐Aryloxythiazol‐5‐yl)but‐3‐yn‐2‐yl)benzamides
Author(s) -
Zhu Youquan,
Liu Pei,
Wang Danyang,
Zhang Jin,
Cheng Jie,
Ma Yuan,
Zou Xiaomao,
Yang Huazheng
Publication year - 2013
Publication title -
chinese journal of chemistry
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 1.28
H-Index - 41
eISSN - 1614-7065
pISSN - 1001-604X
DOI - 10.1002/cjoc.201200824
Subject(s) - chemistry , benzamide , sclerotinia sclerotiorum , bioassay , stereochemistry , proton nmr , elemental analysis , medicinal chemistry , organic chemistry , botany , biology , genetics
A series of novel N ‐(4‐(2‐aryloxythiazol‐5‐yl)but‐3‐yn‐2‐yl)benzamide derivatives were designed and synthesized. Their structures were identified by 1 H NMR and elemental analyses. Preliminary bioassays indicated that some title compounds provided >80% control of Sclerotinia sclerotiorum at 50 µg/mL and >70% herbicidal activities against B. campestris at 100 µg/mL. Their structure‐activities relationships were also discussed.