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Inside Cover: Long Residence Times Revealed by Aurora A Kinase‐Targeting Fluorescent Probes Derived from Inhibitors MLN8237 and VX‐689 (ChemBioChem 3/2014)
Author(s) -
Lavogina Darja,
Enkvist Erki,
Viht Kaido,
Uri Asko
Publication year - 2014
Publication title -
chembiochem
Language(s) - English
Resource type - Reports
SCImago Journal Rank - 1.05
H-Index - 126
eISSN - 1439-7633
pISSN - 1439-4227
DOI - 10.1002/cbic.201490005
Subject(s) - fluorescence , cover (algebra) , chemistry , kinase , dissociation (chemistry) , biophysics , microbiology and biotechnology , biochemistry , biology , physics , organic chemistry , mechanical engineering , quantum mechanics , engineering
The inside cover picture shows fluorescent probes based on well‐known inhibitors MLN8237 and VX‐689 (MK‐5108) that revealed slow association/dissociation kinetics in inhibition and binding assays with Aurora A kinase. For more details see the paper by D. Lavõgina et al. on p. 443 ff.