Premium
Frontispiece: Activity‐Directed Synthesis with Intermolecular Reactions: Development of a Fragment into a Range of Androgen Receptor Agonists
Author(s) -
Karageorgis George,
Dow Mark,
Aimon Anthony,
Warriner Stuart,
Nelson Adam
Publication year - 2015
Publication title -
angewandte chemie international edition
Language(s) - English
Resource type - Reports
SCImago Journal Rank - 5.831
H-Index - 550
eISSN - 1521-3773
pISSN - 1433-7851
DOI - 10.1002/anie.201584661
Subject(s) - androgen receptor , fragment (logic) , intermolecular force , chemistry , molecule , stereochemistry , combinatorial chemistry , biology , computer science , genetics , organic chemistry , cancer , prostate cancer , programming language
Lead Generation Activity‐directed synthesis (ADS), a novel discovery approach in which bioactive molecules emerge in parallel with associated syntheses, is exploited by A. Nelson, S. Warriner et al. in their Communication on page 13538 ff.