Premium
An Alkyne Diboration/6π‐Electrocyclization Strategy for the Synthesis of Pyridine Boronic Acid Derivatives
Author(s) -
MoraRadó Helena,
Bialy Laurent,
Czechtizky Werngard,
Méndez María,
Harrity Joseph P. A.
Publication year - 2016
Publication title -
angewandte chemie
Language(s) - English
Resource type - Journals
eISSN - 1521-3757
pISSN - 0044-8249
DOI - 10.1002/ange.201601084
Subject(s) - alkyne , boronic acid , pyridine , chemistry , combinatorial chemistry , organic chemistry , catalysis
A new and efficient synthesis of pyridine‐based heteroaromatic boronic acid derivatives is reported through a novel diboration/6π‐electrocyclization strategy. This method delivers a range of functionalized heterocycles from readily available starting materials.