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Direct and Site‐Selective Palladium‐Catalyzed C‐7 Acylation of Indolines with Aldehydes
Author(s) -
Shin Youngmi,
Sharma Satyasheel,
Mishra Neeraj Kumar,
Han Sangil,
Park Jihye,
Oh Hyunji,
Ha Jimin,
Yoo Hyunwu,
Jung Young Hoon,
Kim In Su
Publication year - 2015
Publication title -
advanced synthesis and catalysis
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 1.541
H-Index - 155
eISSN - 1615-4169
pISSN - 1615-4150
DOI - 10.1002/adsc.201400942
Subject(s) - chemistry , acylation , palladium , catalysis , oxidative phosphorylation , combinatorial chemistry , organic chemistry , biochemistry
The palladium‐catalyzed oxidative acylation of indolines at the C‐7 position with aldehydes or alcohols via CH bond activation is described. This protocol represents a facile access to 7‐acylated indolines, which can be readily transformed into 7‐acylated indoles with diverse biological properties.