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Arylthiolation of Arylamine Derivatives with (Arylthio)‐ pyrrolidine‐2,5‐diones
Author(s) -
Tian Hua,
Yang Haijun,
Zhu Changjin,
Fu Hua
Publication year - 2015
Publication title -
advanced synthesis and catalysis
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 1.541
H-Index - 155
eISSN - 1615-4169
pISSN - 1615-4150
DOI - 10.1002/adsc.201400929
Subject(s) - chemistry , pyrrolidine , reagent , aryl , catalysis , acetonitrile , combinatorial chemistry , solvent , organic chemistry , alkyl
A simple and efficient method for arylthiolation of arylamines has been developed. The protocol uses (arylthio)pyrrolidine‐2,5‐diones as the arylthiolating reagents, acetonitrile as the solvent, and no catalyst and additive are required, which avoids contamination from the transition metal catalysts in the target products. Therefore, the present method should provide a convenient, efficient and practical strategy for the synthesis of other aryl sulfides.