Exploring kinase inhibition properties of 9<em>H</em>-pyrimido[5,4-<em>b</em>]- and [4,5-<em>b</em>]indol-4-amine derivatives
Author(s) -
Thierry Besson,
Pascal Marchand,
Yvonnick Loidreau,
Carole DubouilhBenard,
MarieRenée Nourrisson,
Nadège Loaëc,
Laurent Meijer
Publication year - 2020
Publication title -
proceedings of 7th international electronic conference on medicinal chemistry
Language(s) - English
Resource type - Conference proceedings
DOI - 10.3390/ecmc2020-07390
Subject(s) - dyrk1a , chemistry , kinase , stereochemistry , ic50 , adenosine kinase , protein kinase a , harmine , biochemistry , enzyme , biology , pharmacology , in vitro , adenosine deaminase
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