Open AccessEnhancement of Muscimol Binding and Gating by Allosteric Modulators of the GABAAReceptor: Relating Occupancy to State Functions
Author(s) -
Gustav Akk,
Allison L. Germann,
Yusuke Sugasawa,
Spencer R. Pierce,
Alex S. Evers,
Joe Henry Steinbach
Publication year - 2020
Publication title -
molecular pharmacology
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 1.469
H-Index - 198
eISSN - 1521-0111
pISSN - 0026-895X
DOI - 10.1124/mol.120.000066
Subject(s) - muscimol , gabaa receptor , pregnenolone sulfate , allosteric regulation , chemistry , neuroactive steroid , agonist , radioligand , allopregnanolone , gabaergic , receptor , biophysics , stereochemistry , biochemistry , biology
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