Novel oral anti-influenza prodrug candidate AV5075S
Author(s) -
Alexandre V. Ivachtchenko,
Yan A. Ivanenkov,
Oleg D. Mitkin,
Pavel Yamanushkin,
V. Bichko,
Natalia A. Shevkun,
O. V. Mokrushina,
O. O. Nevolina,
Ruben N. Karapetian,
Irina A. Leneva,
I. Т. Fedyakina,
Mark S. Veselov
Publication year - 2014
Publication title -
journal of antimicrobial chemotherapy
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 2.124
H-Index - 194
eISSN - 1460-2091
pISSN - 0305-7453
DOI - 10.1093/jac/dkt507
Subject(s) - prodrug , drug candidate , neuraminidase inhibitor , pharmacokinetics , neuraminidase , pharmacology , in vivo , oseltamivir , virus , potency , influenza a virus , drug , docking (animal) , chemistry , in vitro , biology , virology , biochemistry , medicine , covid-19 , infectious disease (medical specialty) , disease , microbiology and biotechnology , nursing , pathology
Development of a novel drug candidate with improved activity against influenza virus neuraminidase (NA) compared with currently available therapeutics.
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