Activity of capuramycin analogues against Mycobacterium tuberculosis, Mycobacterium avium and Mycobacterium intracellularein vitro and in vivo
Author(s) -
Tetsufumi Koga,
Takashi Fukuoka,
Norio Doi,
Tamako Harasaki,
Harumi Inoue,
Hitoshi Hotoda,
Masayo Kakuta,
Yasunori Muramatsu,
Naotoshi Yamamura,
Misa Hoshi,
Takashi Hirota
Publication year - 2004
Publication title -
journal of antimicrobial chemotherapy
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 2.124
H-Index - 194
eISSN - 1460-2091
pISSN - 0305-7453
DOI - 10.1093/jac/dkh417
Subject(s) - antimycobacterial , microbiology and biotechnology , mycobacterium tuberculosis , mycobacterium , tuberculosis , in vivo , broth microdilution , biology , nontuberculous mycobacteria , rifabutin , in vitro , medicine , antibiotics , minimum inhibitory concentration , clarithromycin , pathology , biochemistry
The antimycobacterial activities of RS-112997, RS-124922 and RS-118641, three capuramycin analogues that inhibit phospho-N-acetylmuramyl-pentapeptide translocase, were tested against clinical isolates of Mycobacterium tuberculosis, Mycobacterium avium and Mycobacterium intracellulare.
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