Characterization of a new series of non-covalent proteasome inhibitors with exquisite potency and selectivity for the 20S β5-subunit
Author(s) -
C. Blackburn,
K. M. Gigstad,
P. Hales,
K. Garcia,
M. Jones,
F. J. Bruzzese,
C. Barrett,
J. X. Liu,
T. A. Soucy,
D. S. Sappal,
N. Bump,
E. J. Olhava,
P. Fleming,
L. R. Dick,
C. Tsu,
M. D. Sintchak,
J. L. Blank
Publication year - 2010
Publication title -
biochemical journal
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 1.706
H-Index - 265
eISSN - 1470-8728
pISSN - 0264-6021
DOI - 10.1042/bj4310433u
Subject(s) - proteasome , covalent bond , peptide , protein subunit , selectivity , potency , chemistry , ubiquitin , biochemistry , sentence , computational biology , stereochemistry , biology , in vitro , gene , computer science , natural language processing , organic chemistry , catalysis
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