Tandem Suzuki-Miyaura Coupling/Acid-Catalyzed Cyclization between Vinyl Ether Boronates and Vinyl Halides: A Concise Approach to Polysubstituted Furans
Author(s) -
Alexey N. Butkevich,
Lieven Meerpoel,
Ian Stansfield,
Patrick Angibaud,
Andrei Corbu,
Janine Cossy
Publication year - 2013
Publication title -
organic letters
Language(s) - English
Resource type - Journals
SCImago Journal Rank - 1.94
H-Index - 239
eISSN - 1523-7060
pISSN - 1523-7052
DOI - 10.1021/ol4014574
Subject(s) - chemistry , tandem , dihydropyran , pinacol , catalysis , halide , organic chemistry , boronic acid , coupling (piping) , combinatorial chemistry , mechanical engineering , materials science , engineering , composite material
Polysubstituted 2-(ω-hydroxyalkyl)furans were prepared by tandem Suzuki-Miyaura coupling/acid-catalyzed cyclization starting from appropriately substituted 3-haloallylic alcohols and dihydrofuran-, dihydropyran- or glycal-derived pinacol boronates.
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