Arylation and Heteroarylation of Thienylsulfonamides with Organotrifluoroborates | Zendy

Mnaza Noreen | Zendy; Nasır Rasool | Zendy; Mirna El Khatib | Zendy; Gary A. Molander | Zendy

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Arylation and Heteroarylation of Thienylsulfonamides with Organotrifluoroborates

Author(s) -

Mnaza Noreen,

Nasır Rasool,

Mirna El Khatib,

Gary A. Molander

Publication year - 2014

Publication title -

the journal of organic chemistry

Language(s) - English

Resource type - Journals

SCImago Journal Rank - 1.2

H-Index - 228

eISSN - 1520-6904

pISSN - 0022-3263

DOI - 10.1021/jo501323z

Subject(s) - chemistry , sulfonamide , combinatorial chemistry , suzuki reaction , organic chemistry , aryl , alkyl

A mild, practical protocol has been developed for the Suzuki cross-coupling of unprotected thienylsulfonamides from air- and bench-stable organotrifluoroborates in the absence of a protecting group on the sulfonamide nitrogen. The developed synthetic method can be applied to the preparation of various arylated and heteroarylated thienylsulfonamides under conditions that are tolerant of a broad range of functional groups.

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